Daawada Lacosamide
Magaca Alaabta: Durida Lacosamide
Tilmaamaha:
Lacosamide waa dawo cusub oo jiilka saddexaad ah oo ka hortagta suuxdinta oo loo tilmaamay daawaynta suuxdinta (sida caadiga ah daawaynta isku xidhka ah ee suuxdinta qayb-bilawga ah ee dadka waaweyn iyo dhalinyarada).
Farmaajada Farmaajo:
Lacosamide waxay si xushmad leh u wanaajisaa firfircoonida gaabiska ah ee kanaalada sodium-ka-gated, taas oo dejisa xuubabka neuronal-ka hyperexcitable waxayna joojisaa rasaasta neerfaha ee soo noqnoqda.
Cilmi-baaristu waxay soo jeedinaysaa in lacosamide ay sidoo kale samayn karto saameynteeda anticonvulsant iyada oo loo marayo isdhexgalka dhexdhexaadiyaha jawaab-celinta borotiinka-2 (CRMP-2), oo ah dariiqa ku lug leh calaamadaha neuronal iyo koritaanka axonal.
Waxaa xusid mudan, lacosamide ma saameynayso firfircoonida degdega ah ee kanaalada soodiyamka, taas oo gacan ka geysata yaraynta saamaynta xun ee shaqada maskaxda ee caadiga ah waxayna yaraynaysaa halista neurotoxicity.